Overview of drug transporter families / Guofeng You and Marilyn E. Morris -- Organic Cation and Zwitterion transporters / Megan L. Koleske, Xiaomin Liang, Osatohanmwen Jessica Enogieru, Dina Buitrago, and Kathleen M. Giacomini -- Multidrug and toxin extrusion proteins / Lauren M. Aleksunes, Victoria Woo, and Melanie S. Joy -- Organic anion transporters (OATs) / Jeffry C. Granados, Jingui Zhang, Guofeng You, Sanjay K. Nigam -- Organic anion transporting polypeptides OATP / Rommel G. Tirona and Richard B. Kim -- Mammalian oligopeptide transporters / Stephen M. Carl, Dea Herrera-Ruiz, Rajinder K. Bhardwaj, Olafur Gudmundsson, Stephanie Mowery, and Gregory T. Knipp -- Monocarboxylic acid transporters / Marilyn E. Morris and Nisha V. Kwatra -- The nucleoside transporters CNTs and ENTs / Raj Govindarajan, Antonio López Quiñones, and Joanne Wang -- Bile acid transporters / Ebehiremen N. Ayewoh and Peter W. Swaan -- The P-glycoprotein multidrug transporter / Andaleeb Sajid, Sabrina Lusvarghi and Suresh V. Ambudkar -- Multidrug resistance proteins of the ABCC subfamily / Anne T. Nies and Franziska Klein -- ABCG2, the breast cancer resistance protein (BCRP) / Robert W. Robey, Sabrina Lusvarghi, Cindy H. Chau, Agnes Basseville, William D. Figg, Suresh V. Ambudkar, and Susan E. Bates -- Drug transport in the liver / Noora Sjöstedt, Jeffry Adiwidjaja, William A. Murphy, and Kim L.R. Brouwer -- Drug transport in the brain / Vishal Sangha, Erica I. Williams, Patrick T. Ronaldson, and Reina Bendayan -- Drug transport in the kidney / Douglas H. Sweet -- Drug transporters in the human intestine / Stefan Oswald -- Drug transport in the placenta / Qingcheng Mao, Vadivel Ganapathy, and Jashvant D. Unadkat -- Polymorphisms of drug transporters and clinical relevance / Tore B. Stage and Deanna L. Kroetz -- Ontogeny of drug transporters / Melanie A. Felmlee and Qing Zhang -- Experimental approaches for studying drug transporters / Yusuke Masuo, Azusa Futatsugi, and Yukio Kato -- Transporters mediated drug disposition : physiochemistry and in silico approaches / Manthena V. S. Varma, Ayman El-Kattan, and Yurong Lai -- In vitro-in vivo scale-up of drug transport activities / Kazuya Maeda and Yuichi Sugiyama -- Application of physiologically based pharmacokinetic and pharmacodynamic (PBPK/PD) modeling comprising transporters : delineating the role of various factors in drug disposition and toxicity / Matthew D. Harwood, Amin Rostami-Hodjegan, and Sibylle Neuhoff -- Transporters as therapeutic targets in human diseases / Robert S. Jones and Eugene C. Chen -- Diet/nutrient interactions with drug transporters / Marilyn E. Morris and Tianjing Ren.